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Mohr, Klaus; Prilla, S.; Schrobang, J.; Ellis, J.; Höltje, H.D.: Allosteric interactions with muscarinic acetylcholine receptors: complex role of the conserved tryptophan M2422Trp in a critical cluster of amino acids for baseline affinity, subtype selectivity, and cooperativity. In: Molecular Pharmacology, 70(1), 2006, S. 181-193

Mohr, Klaus; Jäger, D.; Schmalenbach, C.; Prilla, S.; Schrobang, J.; Kebig, A.; Sennwitz, M.; Heller, E.; Tränkle, C.; Holzgrabe, U.; Höltje, H.D.: Allosteric small molecules unveil a role of an extracellular E2/transmembrane helix 7 junction for G protein-coupled receptor activation. In: The Journal of Biological Chemistry, 282(48), 2007, S. 34968-34976

Mohr, Klaus; Antony, J.; Kellershohn, K.; Mohr-Andrä, M.; Kebig, A.; Prilla, S.; Muth, M.; Heller, E.; Disingrini, T.; Dallanoce, C.; Bertoni, S.; Schrobang, J.; Tränkle, C.; Kostenis, E.; Christopoulos, A.; Höltje, H.D.; Barocelli, E.; De Amici, M.; Holzgrabe, U.: Dualsteric GPCR targeting: a novel route to binding and signaling pathway selectivity. In: The Journal of the Federation of American Societies for Experimental Biology, 23(2), 2009, S. 442-450

Mohr, Klaus; Tränkle, C.; Kostenis, E.; Barocelli, E.; De Amici, M.; Holzgrabe, U.: Rational design of dualsteric GPCR ligands: quests and promise. In: British Journal of Pharmacology, 159(5), 2010, S. 997-1008

Mohr, Klaus; Schröder, R.; Janssen, N.; Schmidt, J.; Kebig, A.; Merten, N.; Hennen, S.; Müller, A.; Blättermann, S.; Mohr-Andrä, M.; Zahn, S.; Wenzel, J.; Smith, N.J.; Gomeza, J.; Drewke, C.; Milligan, G.; Kostenis, E.: Deconvolution of complex G protein-coupled receptor signaling in live cells using dynamic mass redistribution measurements. In: Nature Biotechnology, 28(9), 2010, S. 943-949